# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4476817 | BI-0314 | deltaTm | = | 1.4 | degrees C | ALA4309968 | degrees C | ||||
2. | ALA4476817 | BI-0314 | Ratio | = | 650 | /M/s | ALA4309967 | /M/s | Homo sapiens | |||
3. | ALA4476817 | BI-0314 | Kcat | = | 0.042 | /s | ALA4309966 | /s | Homo sapiens | |||
4. | ALA4476817 | BI-0314 | Km | = | 65.4 | uM | ALA4309965 | nM | Homo sapiens | |||
5. | ALA4476817 | BI-0314 | Activity | 0 | ALA4309964 | Active | Mus musculus | |||||
6. | ALA4476817 | BI-0314 | Activity | 0 | ALA4309963 | Not Active | Homo sapiens | |||||
7. | ALA4476817 | BI-0314 | Activity | 0 | ALA4309962 | Not Active | Homo sapiens | |||||
8. | ALA4476817 | BI-0314 | Activity | 0 | ALA4309961 | Not Active | Homo sapiens | |||||
9. | ALA4476817 | BI-0314 | Activity | = | 27 | % | ALA4309960 | % | ||||
10. | ALA4476817 | BI-0314 | Activity | = | 48 | % | ALA4309959 | % | ||||
11. | ALA4476817 | BI-0314 | Activity | = | 61 | % | ALA4309958 | % | Homo sapiens | |||
12. | ALA4476817 | BI-0314 | Activity | = | 28 | % | ALA4309957 | % | ||||
13. | ALA4476817 | BI-0314 | Activity | 0 | ALA4309956 | Dose-dependent effect | ||||||
14. | ALA4476817 | BI-0314 | Activity | = | 33 | % | ALA4309955 | % | ||||
15. | ALA4476817 | BI-0314 | Activity | = | 56 | % | ALA4309954 | % | ||||
16. | ALA4476817 | BI-0314 | Activity | 0 | ALA4309950 | Not Active | Homo sapiens | |||||
17. | ALA4476817 | BI-0314 | Kd | = | 800 | uM | ALA4309949 | 3.10 | nM | Homo sapiens | ||
18. | ALA4476817 | BI-0314 | Kd | = | 38 | uM | ALA4309948 | 4.42 | nM | Homo sapiens | ||
19. | ALA4476817 | BI-0314 | Activity | 0 | ALA4309946 | Active | Homo sapiens |