| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4476839 | 28 | F | = | 60.5 | % | ALA4355768 | % | ||||
| 2. | ALA4476839 | 28 | Vdss | = | 0.85 | L/Kg | ALA4355766 | L.kg-1 | ||||
| 3. | ALA4476839 | 28 | t1/2 | = | 1.18 | hr | ALA4355763 | hr | ||||
| 4. | ALA4476839 | 28 | CL | = | 14.4 | ml/min.kg | ALA4355761 | mL.min-1.kg-1 | ||||
| 5. | ALA4476839 | 28 | AUC/dose | = | 2.96 | uM.hr.kg/mg | ALA4355759 | uM.hr.kg/mg | ||||
| 6. | ALA4476839 | 28 | Fu | > | 99 | % | ALA4355757 | |||||
| 7. | ALA4476839 | 28 | EC50 | = | 328 | nM | ALA4355755 | 6.48 | nM | Rattus norvegicus | ||
| 8. | ALA4476839 | 28 | Ki | = | 35 | nM | ALA4355754 | 7.46 | nM | Homo sapiens | ||
| 9. | ALA4476839 | 28 | Fu | > | 99 | % | ALA4355753 | |||||
| 10. | ALA4476839 | 28 | Papp | = | 26 | 10'-6 cm/s | ALA4355751 | 10'-6 cm/s | ||||
| 11. | ALA4476839 | 28 | Ki | > | 10000 | nM | ALA4355756 | nM | Homo sapiens |
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