| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4483089 | 5 | EC50 | > | 30 | uM | ALA4355805 | nM | Homo sapiens | |||
| 2. | ALA4483089 | 5 | IC50 | > | 50 | uM | ALA4355804 | nM | Homo sapiens | |||
| 3. | ALA4483089 | 5 | IC50 | > | 50 | uM | ALA4355803 | nM | Homo sapiens | |||
| 4. | ALA4483089 | 5 | IC50 | > | 50 | uM | ALA4355802 | nM | Homo sapiens | |||
| 5. | ALA4483089 | 5 | IC50 | > | 30 | uM | ALA4355801 | nM | Homo sapiens | |||
| 6. | ALA4483089 | 5 | IC50 | > | 30 | uM | ALA4355800 | nM | Homo sapiens | |||
| 7. | ALA4483089 | 5 | IC50 | > | 30 | uM | ALA4355799 | nM | Homo sapiens | |||
| 8. | ALA4483089 | 5 | F | = | 62 | % | ALA4355767 | % | ||||
| 9. | ALA4483089 | 5 | Vdss | = | 5.39 | L/Kg | ALA4355764 | L.kg-1 | ||||
| 10. | ALA4483089 | 5 | t1/2 | = | 1.89 | hr | ALA4355762 | hr | ||||
| 11. | ALA4483089 | 5 | CL | = | 66.3 | ml/min.kg | ALA4355760 | mL.min-1.kg-1 | ||||
| 12. | ALA4483089 | 5 | AUC/dose | = | 0.598 | uM.hr.kg/mg | ALA4355758 | uM.hr.kg/mg | ||||
| 13. | ALA4483089 | 5 | Ki | = | 3600 | nM | ALA4355756 | 5.44 | nM | Homo sapiens | ||
| 14. | ALA4483089 | 5 | EC50 | = | 36.7 | nM | ALA4355755 | 7.43 | nM | Rattus norvegicus | ||
| 15. | ALA4483089 | 5 | Ki | = | 5.5 | nM | ALA4355754 | 8.26 | nM | Homo sapiens | ||
| 16. | ALA4483089 | 5 | Papp | = | 1.1 | 10'-6 cm/s | ALA4355751 | 10'-6 cm/s |
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