| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4483477 | 17 | F | = | 3 | % | ALA4359959 | % | ||||
| 2. | ALA4483477 | 17 | AUC | = | 0.5 | uM.hr | ALA4359955 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 3. | ALA4483477 | 17 | Cmax | = | 0.2 | uM | ALA4359951 | nM | ||||
| 4. | ALA4483477 | 17 | Vdss | = | 0.4 | L/Kg | ALA4359950 | L.kg-1 | ||||
| 5. | ALA4483477 | 17 | CL | = | 23 | ml/min.kg | ALA4359949 | mL.min-1.kg-1 | ||||
| 6. | ALA4483477 | 17 | PPB | = | 95 | % | ALA4359948 | % | ||||
| 7. | ALA4483477 | 17 | PPB | = | 88 | % | ALA4359947 | % | ||||
| 8. | ALA4483477 | 17 | Papp | = | 2.4 | 10'-6 cm/s | ALA4359946 | 10'-6 cm/s | ||||
| 9. | ALA4483477 | 17 | IC50 | = | 97 | nM | ALA4359943 | 7.01 | nM | Homo sapiens | ||
| 10. | ALA4483477 | 17 | Ki | > | 6100 | nM | ALA4359941 | nM | Homo sapiens | |||
| 11. | ALA4483477 | 17 | Ki | = | 1.8 | nM | ALA4359940 | 8.74 | nM | Homo sapiens |
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