| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4483512 | 59 | Ratio | > | 4.7 | ALA4392470 | ||||||
| 2. | ALA4483512 | 59 | Papp | = | 71 | nm/s | ALA4392469 | nm/s | ||||
| 3. | ALA4483512 | 59 | Papp | < | 15 | nm/s | ALA4392468 | nm/s | ||||
| 4. | ALA4483512 | 59 | AUClast | = | 75 | nM.hr | ALA4392400 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 5. | ALA4483512 | 59 | Tmax | = | 0.3 | hr | ALA4392399 | hr | ||||
| 6. | ALA4483512 | 59 | Cmax | = | 63 | nM | ALA4392398 | nM | ||||
| 7. | ALA4483512 | 59 | Ratio | = | 0.73 | ALA4392396 | ||||||
| 8. | ALA4483512 | 59 | FC | = | 0.46 | ALA4392395 | ||||||
| 9. | ALA4483512 | 59 | AUClast | = | 27 | % | ALA4392394 | % | ||||
| 10. | ALA4483512 | 59 | AUClast | = | 103 | nM.hr | ALA4392393 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 11. | ALA4483512 | 59 | Tmax | = | 0.4 | hr | ALA4392391 | hr | ||||
| 12. | ALA4483512 | 59 | Cmax | = | 99 | nM | ALA4392389 | nM | ||||
| 13. | ALA4483512 | 59 | solubility | = | 0.009 | mg/ml | ALA4392383 | ug.mL-1 | ||||
| 14. | ALA4483512 | 59 | t1/2 | = | 214.9 | hr | ALA4392382 | hr | ||||
| 15. | ALA4483512 | 59 | solubility | > | 1.42 | mg/ml | ALA4392376 | ug.mL-1 | ||||
| 16. | ALA4483512 | 59 | solubility | > | 0.98 | mg/ml | ALA4392375 | ug.mL-1 | ||||
| 17. | ALA4483512 | 59 | t1/2 | = | 376.3 | hr | ALA4392373 | hr | ||||
| 18. | ALA4483512 | 59 | t1/2 | > | 500 | hr | ALA4392372 | hr |
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