| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4513418 | 7 | Ki | = | 204 | nM | ALA4410512 | 6.69 | nM | Homo sapiens | ||
| 2. | ALA4513418 | 7 | IC50 | > | 100 | uM | ALA4410522 | nM | Homo sapiens | |||
| 3. | ALA4513418 | 7 | IC50 | > | 100 | uM | ALA4410523 | nM | Homo sapiens | |||
| 4. | ALA4513418 | 7 | IC50 | = | 58.5 | uM | ALA4410524 | 4.23 | nM | Homo sapiens | ||
| 5. | ALA4513418 | 7 | IC50 | > | 100 | uM | ALA4410525 | nM | Homo sapiens | |||
| 6. | ALA4513418 | 7 | Activity | 0 | ALA4410533 | Non-Toxic | Rattus norvegicus | |||||
| 7. | ALA4513418 | 7 | Activity | 0 | ALA4410534 | Non-Toxic | Rattus norvegicus | |||||
| 8. | ALA4513418 | 7 | INH | 0 | ALA4410535 | Active | % | Homo sapiens | ||||
| 9. | ALA4513418 | 7 | CL | = | 49.7 | ml/min.kg | ALA4739550 | mL.min-1.kg-1 | ||||
| 10. | ALA4513418 | 7 | CL | = | 29.2 | ml/min.kg | ALA4739549 | mL.min-1.kg-1 | ||||
| 11. | ALA4513418 | 7 | Drugexcretion | = | 36.4 | % | ALA4739548 | % | ||||
| 12. | ALA4513418 | 7 | Vdss | = | 5.2 | L/Kg | ALA4739547 | L.kg-1 | ||||
| 13. | ALA4513418 | 7 | CL | = | 78.9 | ml/min.kg | ALA4739546 | mL.min-1.kg-1 | ||||
| 14. | ALA4513418 | 7 | Ratio | = | 0.7 | ALA4739545 | ||||||
| 15. | ALA4513418 | 7 | AUC | = | 3.2 | uM.hr | ALA4739544 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 16. | ALA4513418 | 7 | Vdss | = | 3.4 | L/Kg | ALA4739543 | L.kg-1 | ||||
| 17. | ALA4513418 | 7 | CL | = | 51.3 | ml/min.kg | ALA4739542 | mL.min-1.kg-1 | ||||
| 18. | ALA4513418 | 7 | t1/2 | = | 6.7 | hr | ALA4739541 | hr | ||||
| 19. | ALA4513418 | 7 | F | = | 0.81 | % | ALA4739519 | % | ||||
| 20. | ALA4513418 | 7 | Vdss | = | 0.7 | L/Kg | ALA4739497 | L.kg-1 |
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