# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4513808 | 14, Single Atropisomer | Activity | = | 50 | % | ALA4324506 | % | Rattus norvegicus | |||
2. | ALA4513808 | 14, Single Atropisomer | Activity | 0 | ALA4324505 | Dose-dependent effect | Rattus norvegicus | |||||
3. | ALA4513808 | 14, Single Atropisomer | Activity | 0 | ALA4324504 | Dose-dependent effect | Rattus norvegicus | |||||
4. | ALA4513808 | 14, Single Atropisomer | Activity | 0 | ALA4324503 | Not Active | Rattus norvegicus | |||||
5. | ALA4513808 | 14, Single Atropisomer | K | = | 0.005 | /min | ALA4324502 | /min | Homo sapiens | |||
6. | ALA4513808 | 14, Single Atropisomer | IC50 | = | 151 | nM | ALA4324501 | 6.82 | nM | Homo sapiens | ||
7. | ALA4513808 | 14, Single Atropisomer | IC50 | > | 10 | uM | ALA4324500 | nM | Homo sapiens | |||
8. | ALA4513808 | 14, Single Atropisomer | IC50 | > | 10 | uM | ALA4324499 | nM | Homo sapiens | |||
9. | ALA4513808 | 14, Single Atropisomer | IC50 | > | 10 | uM | ALA4324498 | nM | Homo sapiens | |||
10. | ALA4513808 | 14, Single Atropisomer | IC50 | > | 10 | uM | ALA4324497 | nM | Homo sapiens | |||
11. | ALA4513808 | 14, Single Atropisomer | IC50 | > | 10 | uM | ALA4324496 | nM | Homo sapiens | |||
12. | ALA4513808 | 14, Single Atropisomer | IC50 | > | 10 | uM | ALA4324495 | nM | Homo sapiens | |||
13. | ALA4513808 | 14, Single Atropisomer | IC50 | > | 10 | uM | ALA4324494 | nM | Homo sapiens | |||
14. | ALA4513808 | 14, Single Atropisomer | IC50 | > | 10 | uM | ALA4324493 | nM | Homo sapiens | |||
15. | ALA4513808 | 14, Single Atropisomer | IC50 | > | 10 | uM | ALA4324492 | nM | Homo sapiens | |||
16. | ALA4513808 | 14, Single Atropisomer | IC50 | > | 10 | uM | ALA4324491 | nM | Homo sapiens | |||
17. | ALA4513808 | 14, Single Atropisomer | IC50 | = | 151 | nM | ALA4324490 | 6.82 | nM | Homo sapiens | ||
18. | ALA4513808 | 14, Single Atropisomer | Tmax | = | 1 | hr | ALA4324489 | hr | ||||
19. | ALA4513808 | 14, Single Atropisomer | Cmax/dose | = | 2448 | nM | ALA4324488 | nM | ||||
20. | ALA4513808 | 14, Single Atropisomer | F | = | 90 | % | ALA4324487 | % |