| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4515137 | 16 | CLH | = | 48 | ml/min.kg | ALA5236799 | mL.min-1.kg-1 | ||||
| 2. | ALA4515137 | 16 | Activity | = | 15 | % | ALA5236793 | % | Homo sapiens | |||
| 3. | ALA4515137 | 16 | F | = | 63 | % | ALA5236792 | % | ||||
| 4. | ALA4515137 | 16 | t1/2 | = | 3.7 | hr | ALA5236791 | hr | ||||
| 5. | ALA4515137 | 16 | EC50 | = | 49 | nM | ALA5236783 | 7.31 | nM | Homo sapiens | ||
| 6. | ALA4515137 | 16 | CLH | = | 112 | ml/min.kg | ALA5236777 | mL.min-1.kg-1 | ||||
| 7. | ALA4515137 | 16 | IC50 | = | 81 | nM | ALA5236775 | 7.09 | nM | Homo sapiens | ||
| 8. | ALA4515137 | 16 | CL free | = | 319 | ml/min.kg | ALA4410882 | mL.min-1.kg-1 | ||||
| 9. | ALA4515137 | 16 | Ratio | = | 1 | ALA4410883 | Homo sapiens | |||||
| 10. | ALA4515137 | 16 | IC90 | = | 1215 | nM | ALA4410848 | nM | Homo sapiens | |||
| 11. | ALA4515137 | 16 | IC50 | = | 59 | nM | ALA4410880 | 7.23 | nM | Rattus norvegicus | ||
| 12. | ALA4515137 | 16 | IC50 | = | 28 | nM | ALA4410881 | 7.55 | nM | Mus musculus | ||
| 13. | ALA4515137 | 16 | Activity | = | 79 | % | ALA4410879 | % | Mus musculus | |||
| 14. | ALA4515137 | 16 | Activity | = | 15 | % | ALA4410878 | % | Mus musculus | |||
| 15. | ALA4515137 | 16 | Stability | = | 77.1 | % | ALA4410877 | % | ||||
| 16. | ALA4515137 | 16 | Stability | = | 97 | % | ALA4410875 | % | ||||
| 17. | ALA4515137 | 16 | Stability | = | 81.5 | % | ALA4410876 | % | ||||
| 18. | ALA4515137 | 16 | Stability | 0 | ALA4410874 | Not Determined | % | |||||
| 19. | ALA4515137 | 16 | Stability | = | 96.2 | % | ALA4410873 | % | ||||
| 20. | ALA4515137 | 16 | Stability | 0 | ALA4410872 | Not Determined | % |
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