| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4516240 | 5B | Ke | = | 15 | nM | ALA4433516 | nM | Rattus norvegicus | |||
| 2. | ALA4516240 | 5B | Activity | = | 100 | % | ALA4433515 | % | Rattus norvegicus | |||
| 3. | ALA4516240 | 5B | logP | = | 5.8 | ALA4433514 | ||||||
| 4. | ALA4516240 | 5B | Time | = | 150 | min | ALA4433513 | hr | Mus musculus | |||
| 5. | ALA4516240 | 5B | MPE | = | 100 | % | ALA4433507 | % | Mus musculus | |||
| 6. | ALA4516240 | 5B | Efficacy | 0 | ALA4433505 | Not Active | Homo sapiens | |||||
| 7. | ALA4516240 | 5B | Efficacy | 0 | ALA4433502 | Not Active | Rattus norvegicus | |||||
| 8. | ALA4516240 | 5B | Efficacy | = | 57 | % | ALA4433503 | % | Rattus norvegicus | |||
| 9. | ALA4516240 | 5B | EC50 | 0 | ALA4433504 | Not Active | Homo sapiens | |||||
| 10. | ALA4516240 | 5B | EC50 | 0 | ALA4433506 | Not Active | Rattus norvegicus | |||||
| 11. | ALA4516240 | 5B | EC50 | = | 7.9 | nM | ALA4433508 | 8.10 | nM | Rattus norvegicus | ||
| 12. | ALA4516240 | 5B | Ratio Ki | = | 2 | ALA4433509 | ||||||
| 13. | ALA4516240 | 5B | Ki | = | 160 | nM | ALA4433510 | 6.80 | nM | Homo sapiens | ||
| 14. | ALA4516240 | 5B | Ki | = | 0.46 | nM | ALA4433511 | 9.34 | nM | Rattus norvegicus | ||
| 15. | ALA4516240 | 5B | Ki | = | 0.26 | nM | ALA4433512 | 9.59 | nM | Rattus norvegicus |
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