# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4517711 | 9b | TGI | 0 | ALA4386059 | Not Active | Homo sapiens | |||||
2. | ALA4517711 | 9b | TGI | 0 | ALA4386058 | Not Active | Homo sapiens | |||||
3. | ALA4517711 | 9b | IC50 | > | 1000 | nM | ALA4386056 | nM | Homo sapiens | |||
4. | ALA4517711 | 9b | IC50 | > | 1000 | nM | ALA4386055 | nM | Homo sapiens | |||
5. | ALA4517711 | 9b | Ratio IC50 | > | 100 | ALA4386061 | Homo sapiens | |||||
6. | ALA4517711 | 9b | F | = | 22.5 | % | ALA4385979 | % | ||||
7. | ALA4517711 | 9b | CL | = | 0.89 | L/kg/hr | ALA4385978 | mL.min-1.kg-1 | ||||
8. | ALA4517711 | 9b | beta t1/2 | = | 6.22 | hr | ALA4385977 | hr | ||||
9. | ALA4517711 | 9b | Tmax | = | 0.28 | hr | ALA4385976 | hr | ||||
10. | ALA4517711 | 9b | IC50 | = | 4.83 | nM | ALA4385975 | 8.32 | nM | Mus musculus | ||
11. | ALA4517711 | 9b | IC50 | = | 2.35 | nM | ALA4385974 | 8.63 | nM | Mus musculus | ||
12. | ALA4517711 | 9b | IC50 | = | 0.16 | nM | ALA4385973 | 9.80 | nM | Mus musculus | ||
13. | ALA4517711 | 9b | IC50 | = | 6 | nM | ALA4385972 | 8.22 | nM | Homo sapiens | ||
14. | ALA4517711 | 9b | IC50 | = | 0.043 | nM | ALA4385970 | 10.37 | nM | Homo sapiens | ||
15. | ALA4517711 | 9b | IC50 | < | 0.001 | nM | ALA4385971 | nM | Homo sapiens |