# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4521141 | IIIb | pIC50 | = | 1.71 | ALA4347002 | nM | Homo sapiens | ||||
2. | ALA4521141 | IIIb | IC50 | = | 0.18 | uM | ALA4347002 | 6.75 | nM | Homo sapiens | ||
3. | ALA4521141 | IIIb | FC | = | 2.51 | ALA4347020 | Homo sapiens | |||||
4. | ALA4521141 | IIIb | FC | = | 2.38 | ALA4347021 | Homo sapiens | |||||
5. | ALA4521141 | IIIb | FC | = | 1.06 | ALA4347022 | Homo sapiens | |||||
6. | ALA4521141 | IIIb | FC | = | 0.91 | ALA4347023 | Homo sapiens | |||||
7. | ALA4521141 | IIIb | Activity | 0 | ALA4347019 | Active | ||||||
8. | ALA4521141 | IIIb | Activity | 0 | ALA4347018 | Active | ||||||
9. | ALA4521141 | IIIb | FC | = | 0.6 | ALA4347017 | ||||||
10. | ALA4521141 | IIIb | INH | = | 59.2 | % | ALA4347016 | % | ||||
11. | ALA4521141 | IIIb | FC | = | 0.6 | ALA4347015 | ||||||
12. | ALA4521141 | IIIb | INH | = | 51.9 | % | ALA4347014 | % | ||||
13. | ALA4521141 | IIIb | Activity | = | 4 | % | ALA4347013 | % | ||||
14. | ALA4521141 | IIIb | Activity | = | 17.3 | % | ALA4347012 | % | ||||
15. | ALA4521141 | IIIb | Activity | = | 41 | % | ALA4347011 | % | ||||
16. | ALA4521141 | IIIb | Activity | = | 63.7 | % | ALA4347010 | % | ||||
17. | ALA4521141 | IIIb | Activity | = | 92.7 | % | ALA4347009 | % | ||||
18. | ALA4521141 | IIIb | Selectivity Index | = | 43 | ALA4346949 | ||||||
19. | ALA4521141 | IIIb | IC50 | = | 12.9 | uM | ALA4346948 | 4.89 | nM | Homo sapiens |