# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4521319 | 4A | logP | = | 3.3 | ALA4433514 | ||||||
2. | ALA4521319 | 4A | Time | = | 60 | min | ALA4433513 | hr | Mus musculus | |||
3. | ALA4521319 | 4A | MPE | = | 100 | % | ALA4433507 | % | Mus musculus | |||
4. | ALA4521319 | 4A | Efficacy | = | 60 | % | ALA4433505 | % | Homo sapiens | |||
5. | ALA4521319 | 4A | Efficacy | = | 22 | % | ALA4433502 | % | Rattus norvegicus | |||
6. | ALA4521319 | 4A | Efficacy | = | 98 | % | ALA4433503 | % | Rattus norvegicus | |||
7. | ALA4521319 | 4A | EC50 | = | 121 | nM | ALA4433504 | 6.92 | nM | Homo sapiens | ||
8. | ALA4521319 | 4A | EC50 | = | 12 | nM | ALA4433506 | 7.92 | nM | Rattus norvegicus | ||
9. | ALA4521319 | 4A | EC50 | = | 0.23 | nM | ALA4433508 | 9.64 | nM | Rattus norvegicus | ||
10. | ALA4521319 | 4A | Ratio Ki | = | 7 | ALA4433509 | ||||||
11. | ALA4521319 | 4A | Ki | = | 8 | nM | ALA4433510 | 8.10 | nM | Homo sapiens | ||
12. | ALA4521319 | 4A | Ki | = | 0.41 | nM | ALA4433511 | 9.39 | nM | Rattus norvegicus | ||
13. | ALA4521319 | 4A | Ki | = | 0.06 | nM | ALA4433512 | 10.22 | nM | Rattus norvegicus |