# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4522217 | 25; FM26 | PPB | = | 99.9 | % | ALA5132010 | % | ||||
2. | ALA4522217 | 25; FM26 | Stability | = | 79.1 | % | ALA5132009 | % | ||||
3. | ALA4522217 | 25; FM26 | Stability | = | 73 | % | ALA5132008 | % | ||||
4. | ALA4522217 | 25; FM26 | CLH | = | 31.2 | microL/min/mg | ALA5132007 | mL.min-1.g-1 | ||||
5. | ALA4522217 | 25; FM26 | permeability | = | 36.1 | % | ALA5132006 | % | ||||
6. | ALA4522217 | 25; FM26 | Kinetic_solubility | = | 460 | uM | ALA5132005 | nM | ||||
7. | ALA4522217 | 25; FM26 | INH | = | 0.11 | ALA5132004 | % | |||||
8. | ALA4522217 | 25; FM26 | Selectivity ratio | = | 8 | ALA5132003 | ||||||
9. | ALA4522217 | 25; FM26 | Ratio IC50 | = | 30 | ALA5132002 | ||||||
10. | ALA4522217 | 25; FM26 | deltaTm | = | 0.3 | degrees C | ALA5132001 | degrees C | Homo sapiens | |||
11. | ALA4522217 | 25; FM26 | FC | = | 9.3 | ALA5132000 | ||||||
12. | ALA4522217 | 25; FM26 | deltaTm | = | 2.4 | degrees C | ALA5131999 | degrees C | Homo sapiens | |||
13. | ALA4522217 | 25; FM26 | IC50 | = | 0.1 | uM | ALA5131998 | 7.00 | nM | Homo sapiens | ||
14. | ALA4522217 | 25; FM26 | IC50 | = | 0.27 | uM | ALA5131997 | 6.57 | nM | Homo sapiens | ||
15. | ALA4522217 | 25; FM26 | EC50 | = | 8.2 | uM | ALA5131996 | 5.09 | nM | Homo sapiens | ||
16. | ALA4522217 | 25; FM26 | IC50 | = | 81 | uM | ALA5131995 | 4.09 | nM | Homo sapiens | ||
17. | ALA4522217 | 25; FM26 | Activity | 0 | ALA5129645 | Active | Homo sapiens | |||||
18. | ALA4522217 | 25; FM26 | Activity | 0 | ALA5129644 | NA | Homo sapiens | |||||
19. | ALA4522217 | 25; FM26 | EC50 | = | 330 | nM | ALA5129643 | 6.48 | nM | Homo sapiens | ||
20. | ALA4522217 | 25; FM26 | EC50 | = | 5.6 | uM | ALA5129633 | 5.25 | nM | Homo sapiens |