# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4522605 | 1; KMH-233 | Activity | 0 | ALA4426069 | Active | Homo sapiens | |||||
2. | ALA4522605 | 1; KMH-233 | Activity | 0 | ALA4426068 | Tde | Mus musculus | |||||
3. | ALA4522605 | 1; KMH-233 | Ratio IC50 | = | 6.9 | ALA4426067 | ||||||
4. | ALA4522605 | 1; KMH-233 | Stability | 0 | ALA4426066 | Stable | % | |||||
5. | ALA4522605 | 1; KMH-233 | Cp | = | 0.23 | uM | ALA4426064 | uM | ||||
6. | ALA4522605 | 1; KMH-233 | INH | = | 14 | % | ALA4426063 | % | Mus musculus | |||
7. | ALA4522605 | 1; KMH-233 | Cp | = | 20 | uM | ALA4426062 | uM | ||||
8. | ALA4522605 | 1; KMH-233 | INH | = | 27 | % | ALA4426061 | % | Mus musculus | |||
9. | ALA4522605 | 1; KMH-233 | INH | = | 79 | % | ALA4426060 | % | Mus musculus | |||
10. | ALA4522605 | 1; KMH-233 | Ratio | = | 156 | ALA4426059 | Mus musculus | |||||
11. | ALA4522605 | 1; KMH-233 | Kin | = | 8.2 | 10'-5ml/s/g | ALA4426058 | 10'-5ml/s/g | Mus musculus | |||
12. | ALA4522605 | 1; KMH-233 | Activity | 0 | ALA4426057 | Not Active | Homo sapiens | |||||
13. | ALA4522605 | 1; KMH-233 | beta t1/2 | = | 19.8 | min | ALA4426056 | hr | ||||
14. | ALA4522605 | 1; KMH-233 | beta t1/2 | = | 71.6 | min | ALA4426055 | hr | ||||
15. | ALA4522605 | 1; KMH-233 | beta t1/2 | = | 41.8 | min | ALA4426054 | hr | ||||
16. | ALA4522605 | 1; KMH-233 | beta t1/2 | = | 52.8 | min | ALA4426053 | hr | ||||
17. | ALA4522605 | 1; KMH-233 | beta t1/2 | = | 12 | min | ALA4426052 | hr | ||||
18. | ALA4522605 | 1; KMH-233 | beta t1/2 | = | 44.9 | min | ALA4426051 | hr | ||||
19. | ALA4522605 | 1; KMH-233 | Tmax | = | 30 | min | ALA4426050 | hr | ||||
20. | ALA4522605 | 1; KMH-233 | Tmax | = | 30 | min | ALA4426049 | hr |