| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4522646 | Ex 111 | T/C | = | 0.14 | ALA4421200 | ||||||
| 2. | ALA4522646 | Ex 111 | T/C | = | 0.26 | ALA4421198 | ||||||
| 3. | ALA4522646 | Ex 111 | T/C | = | 0.53 | ALA4421196 | Homo sapiens | |||||
| 4. | ALA4522646 | Ex 111 | F | = | 68 | % | ALA4421193 | % | ||||
| 5. | ALA4522646 | Ex 111 | F | = | 48 | % | ALA4421192 | % | ||||
| 6. | ALA4522646 | Ex 111 | t1/2 | = | 1.3 | hr | ALA4421191 | hr | ||||
| 7. | ALA4522646 | Ex 111 | t1/2 | = | 1.1 | hr | ALA4421190 | hr | ||||
| 8. | ALA4522646 | Ex 111 | Cmax | = | 6.5 | uM | ALA4421189 | nM | ||||
| 9. | ALA4522646 | Ex 111 | Cmax | = | 27 | uM | ALA4421188 | nM | ||||
| 10. | ALA4522646 | Ex 111 | AUC | = | 19 | uM.hr | ALA4421187 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 11. | ALA4522646 | Ex 111 | AUC | = | 18 | uM.hr | ALA4421186 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 12. | ALA4522646 | Ex 111 | IC50 | > | 100 | uM | ALA4421185 | nM | Sus scrofa | |||
| 13. | ALA4522646 | Ex 111 | IC50 | > | 100 | uM | ALA4421184 | nM | Homo sapiens | |||
| 14. | ALA4522646 | Ex 111 | IC50 | > | 100 | uM | ALA4421183 | nM | Homo sapiens | |||
| 15. | ALA4522646 | Ex 111 | IC50 | = | 0.13 | uM | ALA4421182 | 6.89 | nM | Homo sapiens | ||
| 16. | ALA4522646 | Ex 111 | IC50 | = | 0.19 | uM | ALA4421179 | 6.72 | nM | |||
| 17. | ALA4522646 | Ex 111 | IC50 | > | 100 | uM | ALA4421175 | nM |
The page will load shortly, Thanks for your patience!