# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4522782 | 33 | Kinetic_solubility | = | 3.1 | 10'-5mg/ml | ALA4384339 | 10'-5mg/ml | ||||
2. | ALA4522782 | 33 | Kinetic_solubility | = | 4.8 | 10'-5mg/ml | ALA4384338 | 10'-5mg/ml | ||||
3. | ALA4522782 | 33 | CLH | = | 15 | ml/min | ALA4384337 | ml/min | ||||
4. | ALA4522782 | 33 | t1/2 | = | 47 | min | ALA4384336 | hr | ||||
5. | ALA4522782 | 33 | GI50 | > | 10 | uM | ALA4384335 | nM | ||||
6. | ALA4522782 | 33 | EC50 | = | 0.4 | uM | ALA4384334 | 6.40 | nM | Mus musculus | ||
7. | ALA4522782 | 33 | Activity | > | 30000 | % | ALA4384331 | % | Mus musculus | |||
8. | ALA4522782 | 33 | IC50 | = | 0.4 | uM | ALA4384330 | 6.40 | nM | |||
9. | ALA4522782 | 33 | Activity | = | 27000 | % | ALA4384328 | % | Mus musculus | |||
10. | ALA4522782 | 33 | IC50 | = | 1.6 | uM | ALA4384327 | 5.80 | nM | |||
11. | ALA4522782 | 33 | INH | = | 2.9 | % | ALA4384324 | % |