# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4526974 | 1bs | IC50 | = | 15 | nM | ALA4402235 | 7.82 | nM | Homo sapiens | ||
2. | ALA4526974 | 1bs | t1/2 | > | 180 | min | ALA4402237 | hr | ||||
3. | ALA4526974 | 1bs | IC50 | = | 100 | nM | ALA4402238 | 7.00 | nM | Rattus norvegicus | ||
4. | ALA4526974 | 1bs | Papp | = | 470 | nm/s | ALA4402239 | nm/s | ||||
5. | ALA4526974 | 1bs | solubility | = | 0.016 | mg/ml | ALA4402240 | ug.mL-1 | ||||
6. | ALA4526974 | 1bs | beta t1/2 | = | 7.9 | min | ALA4402241 | hr | ||||
7. | ALA4526974 | 1bs | AUC/dose | = | 1900 | ng/hr/ml | ALA4402245 | ng/hr/ml | ||||
8. | ALA4526974 | 1bs | F | = | 46 | % | ALA4402244 | % | ||||
9. | ALA4526974 | 1bs | Vdss | = | 2.5 | L/Kg | ALA4402243 | L.kg-1 | ||||
10. | ALA4526974 | 1bs | CL | = | 3.8 | ml/min.kg | ALA4402242 | mL.min-1.kg-1 |