# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4527241 | 21a | Activity | 0 | ALA4411954 | Dose-dependent effect | ||||||
2. | ALA4527241 | 21a | Activity | 0 | ALA4411949 | Not Active | Rattus norvegicus | |||||
3. | ALA4527241 | 21a | Activity | = | 40 | % | ALA4411944 | % | Rattus norvegicus | |||
4. | ALA4527241 | 21a | Activity | = | 40 | % | ALA4411943 | % | Rattus norvegicus | |||
5. | ALA4527241 | 21a | Activity | 0 | ALA4411942 | Dose-dependent effect | Rattus norvegicus | |||||
6. | ALA4527241 | 21a | Activity | 0 | ALA4411941 | Dose-dependent effect | Rattus norvegicus | |||||
7. | ALA4527241 | 21a | Activity | 0 | ALA4411940 | Active | Rattus norvegicus | |||||
8. | ALA4527241 | 21a | Activity | 0 | ALA4411939 | Active | Mus musculus | |||||
9. | ALA4527241 | 21a | IC50 | < | 3 | uM | ALA4411932 | nM | Homo sapiens | |||
10. | ALA4527241 | 21a | Activity | 0 | ALA4411932 | Dose-dependent effect | Homo sapiens | |||||
11. | ALA4527241 | 21a | CLH | = | 46.22 | ml/min/mg | ALA4411925 | mL.min-1.g-1 | ||||
12. | ALA4527241 | 21a | t1/2 | = | 15 | min | ALA4411924 | hr | ||||
13. | ALA4527241 | 21a | Activity | 0 | ALA4411919 | Active | Homo sapiens | |||||
14. | ALA4527241 | 21a | Activity | = | 61 | % | ALA4411918 | % | ||||
15. | ALA4527241 | 21a | Ki | = | 0.382 | uM | ALA4411915 | 6.42 | nM | Homo sapiens | ||
16. | ALA4527241 | 21a | IC50 | = | 0.126 | uM | ALA4411916 | 6.90 | nM | Homo sapiens | ||
17. | ALA4527241 | 21a | Activity | = | 31 | % | ALA4411917 | % | Homo sapiens |