# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4528928 | 4i | Activity | 0 | ALA4393797 | Non-Toxic | ||||||
2. | ALA4528928 | 4i | Activity | 0 | ALA4393796 | Non-Toxic | ||||||
3. | ALA4528928 | 4i | Activity | 0 | ALA4393795 | Non-Toxic | ||||||
4. | ALA4528928 | 4i | Activity | 0 | ALA4393794 | Non-Toxic | ||||||
5. | ALA4528928 | 4i | Papp | = | 20.5 | 10'-6 cm/s | ALA4393793 | 10'-6 cm/s | ||||
6. | ALA4528928 | 4i | CLH | = | 12.8 | uL/min | ALA4393792 | uL/min | ||||
7. | ALA4528928 | 4i | CLH | = | 4 | uL/min | ALA4393791 | uL/min | ||||
8. | ALA4528928 | 4i | fIC50 | = | 7.4 | nM | ALA4393790 | nM | Homo sapiens | |||
9. | ALA4528928 | 4i | IC50 | = | 59 | nM | ALA4393789 | 7.23 | nM | Homo sapiens | ||
10. | ALA4528928 | 4i | solubility | = | 225 | uM | ALA4393788 | nM | ||||
11. | ALA4528928 | 4i | logD | = | 3.1 | ALA4393787 | ||||||
12. | ALA4528928 | 4i | fpIC50 | = | 8.1 | ALA4351251 | Homo sapiens | |||||
13. | ALA4528928 | 4i | pIC50 | < | 4.6 | ALA4351237 | nM | Homo sapiens | ||||
14. | ALA4528928 | 4i | Selectivity ratio | >= | 100 | ALA4351242 | ||||||
15. | ALA4528928 | 4i | Selectivity ratio | >= | 100 | ALA4351241 | ||||||
16. | ALA4528928 | 4i | INH | 0 | ALA4351239 | Not Active | % | Homo sapiens | ||||
17. | ALA4528928 | 4i | INH | 0 | ALA4351240 | Not Active | % | Homo sapiens | ||||
18. | ALA4528928 | 4i | INH | 0 | ALA4351296 | Not Active | % | Homo sapiens | ||||
19. | ALA4528928 | 4i | INH | 0 | ALA4351295 | Not Active | % | Homo sapiens | ||||
20. | ALA4528928 | 4i | INH | 0 | ALA4351299 | Not Active | % | Homo sapiens |