| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4529950 | 9b | Ratio ED50 | = | 17 | ALA4310633 | Rattus norvegicus | |||||
| 2. | ALA4529950 | 9b | Ratio ED50 | = | 413 | ALA4310632 | ||||||
| 3. | ALA4529950 | 9b | ED50 | = | 16.54 | mg kg-1 | ALA4310631 | mg.kg-1 | Rattus norvegicus | |||
| 4. | ALA4529950 | 9b | ED50 | = | 0.99 | mg kg-1 | ALA4310629 | mg.kg-1 | Rattus norvegicus | |||
| 5. | ALA4529950 | 9b | ED50 | = | 0.04 | mg kg-1 | ALA4310627 | mg.kg-1 | Mustela putorius furo | |||
| 6. | ALA4529950 | 9b | Ke | = | 3.6 | nM | ALA4310626 | nM | Homo sapiens | |||
| 7. | ALA4529950 | 9b | Ke | = | 3.2 | nM | ALA4310625 | nM | Homo sapiens | |||
| 8. | ALA4529950 | 9b | Stability | > | 80 | % | ALA4310624 | % | ||||
| 9. | ALA4529950 | 9b | Stability | 0 | ALA4310623 | Stable | % | |||||
| 10. | ALA4529950 | 9b | Cmax | 0 | ALA4310621 | Not Determined | ||||||
| 11. | ALA4529950 | 9b | F | = | 57 | % | ALA4310619 | % | ||||
| 12. | ALA4529950 | 9b | CL | = | 36 | ml/min.kg | ALA4310618 | mL.min-1.kg-1 | ||||
| 13. | ALA4529950 | 9b | Stability | = | 78 | % | ALA4310617 | % | ||||
| 14. | ALA4529950 | 9b | Stability | = | 89 | % | ALA4310616 | % | ||||
| 15. | ALA4529950 | 9b | Ki | = | 6.8 | nM | ALA4310615 | 8.17 | nM | Homo sapiens | ||
| 16. | ALA4529950 | 9b | Ki | = | 1 | nM | ALA4310614 | 9.00 | nM | Homo sapiens |
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