# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4530951 | 6k | Activity | 0 | ALA4388753 | Active | Rattus norvegicus | |||||
2. | ALA4530951 | 6k | Activity | 0 | ALA4388752 | Active | Rattus norvegicus | |||||
3. | ALA4530951 | 6k | Activity | 0 | ALA4388751 | Active | Rattus norvegicus | |||||
4. | ALA4530951 | 6k | AUC | = | 29.8 | microg.hr/mL | ALA4388748 | ng.hr.mL-1 | ||||
5. | ALA4530951 | 6k | Cmax | = | 10.4 | ug ml-1 | ALA4388747 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
6. | ALA4530951 | 6k | Activity | = | 89 | % | ALA4388737 | % | Homo sapiens | |||
7. | ALA4530951 | 6k | INH | = | 2 | % | ALA4388746 | % | Homo sapiens | |||
8. | ALA4530951 | 6k | INH | = | 0 | % | ALA4388745 | % | Homo sapiens | |||
9. | ALA4530951 | 6k | INH | = | 1 | % | ALA4388744 | % | Homo sapiens | |||
10. | ALA4530951 | 6k | INH | = | 1 | % | ALA4388743 | % | Homo sapiens | |||
11. | ALA4530951 | 6k | INH | = | 11 | % | ALA4388738 | % | Homo sapiens | |||
12. | ALA4530951 | 6k | Stability | = | 85 | % | ALA4388742 | % | ||||
13. | ALA4530951 | 6k | Stability | = | 92 | % | ALA4388741 | % | ||||
14. | ALA4530951 | 6k | solubility | = | 180 | ug ml-1 | ALA4388740 | ug.mL-1 | ||||
15. | ALA4530951 | 6k | EC200 | = | 0.25 | ug ml-1 | ALA4388739 | ug ml-1 | Mus musculus |