# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | CLK-IN-T3 | EUB0000321 | Selectivity ratio | = | 30 | ALA5237414 | ||||||
2. | CLK-IN-T3 | EUB0000321 | INH | 0 | ALA5237386 | Dose-Dependent Effect | % | Homo sapiens | ||||
3. | CLK-IN-T3 | EUB0000321 | IC50 | = | 17 | nM | ALA5237385 | 7.77 | nM | Homo sapiens | ||
4. | CLK-IN-T3 | EUB0000321 | IC50 | = | 0.67 | nM | ALA5237375 | 9.17 | nM | Homo sapiens | ||
5. | CLK-IN-T3 | EUB0000321 | IC50 | = | 110 | nM | ALA5237373 | 6.96 | nM | Homo sapiens | ||
6. | CLK-IN-T3 | EUB0000321 | IC50 | = | 125 | nM | ALA5213242 | 6.90 | nM | Homo sapiens | ||
7. | CLK-IN-T3 | EUB0000321 | % of control | = | 24 | % | ALA5213258 | % | Homo sapiens | |||
8. | CLK-IN-T3 | EUB0000321 | IC50 | = | 3 | uM | ALA5213257 | 5.52 | nM | Homo sapiens | ||
9. | CLK-IN-T3 | EUB0000321 | IC50 | = | 2.52 | uM | ALA5213256 | 5.60 | nM | Homo sapiens | ||
10. | CLK-IN-T3 | EUB0000321 | % of control | = | 29 | % | ALA5213255 | % | Homo sapiens | |||
11. | CLK-IN-T3 | EUB0000321 | IC50 | > | 10 | uM | ALA5213248 | nM | Homo sapiens | |||
12. | CLK-IN-T3 | EUB0000321 | % of control | = | 19 | % | ALA5213247 | % | Homo sapiens | |||
13. | CLK-IN-T3 | EUB0000321 | IC50 | > | 10 | uM | ALA5213250 | nM | Homo sapiens | |||
14. | CLK-IN-T3 | EUB0000321 | % of control | = | 4.9 | % | ALA5213249 | % | Homo sapiens | |||
15. | CLK-IN-T3 | EUB0000321 | IC50 | = | 2.44 | uM | ALA5213254 | 5.61 | nM | Homo sapiens | ||
16. | CLK-IN-T3 | EUB0000321 | % of control | = | 14 | % | ALA5213253 | % | Homo sapiens | |||
17. | CLK-IN-T3 | EUB0000321 | Ki | = | 2154.79 | nM | ALA5213241 | 5.67 | nM | Homo sapiens | ||
18. | CLK-IN-T3 | EUB0000321 | IC50 | = | 138 | uM | ALA5213252 | nM | Homo sapiens | |||
19. | CLK-IN-T3 | EUB0000321 | IC50 | = | 2.44 | uM | ALA5213251 | 5.61 | nM | Homo sapiens | ||
20. | CLK-IN-T3 | EUB0000321 | IC50 | = | 67 | nM | ALA5213244 | 7.17 | nM | Homo sapiens |