# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4534617 | 18.HCl | EC1.5 | = | 30 | uM | ALA4357391 | uM | Oryctolagus cuniculus | |||
2. | ALA4534617 | 18.HCl | Ki | = | 4.6 | nM | ALA4357390 | 8.34 | nM | |||
3. | ALA4534617 | 18.HCl | t1/2 | = | 54 | min | ALA4357330 | hr | ||||
4. | ALA4534617 | 18.HCl | t1/2 | > | 120 | min | ALA4357331 | hr | ||||
5. | ALA4534617 | 18.HCl | t1/2 | > | 120 | min | ALA4357338 | hr | ||||
6. | ALA4534617 | 18.HCl | Ratio | = | 16 | ALA4357337 | ||||||
7. | ALA4534617 | 18.HCl | permeability | = | 348 | nm/s | ALA4357336 | nm/s | ||||
8. | ALA4534617 | 18.HCl | permeability | = | 22 | nm/s | ALA4357335 | nm/s | ||||
9. | ALA4534617 | 18.HCl | t1/2 | = | 81 | min | ALA4357334 | hr | ||||
10. | ALA4534617 | 18.HCl | EC1.5 | = | 1.4 | uM | ALA4357333 | uM | Homo sapiens | |||
11. | ALA4534617 | 18.HCl | Ki | = | 2.2 | nM | ALA4357332 | 8.66 | nM | Homo sapiens |