# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4537527 | 14 | Fu | < | 0.2 | % | ALA4308768 | |||||
2. | ALA4537527 | 14 | Fu | = | 0.4 | % | ALA4308767 | |||||
3. | ALA4537527 | 14 | t1/2 | = | 88 | min | ALA4308766 | hr | ||||
4. | ALA4537527 | 14 | t1/2 | > | 120 | min | ALA4308765 | hr | ||||
5. | ALA4537527 | 14 | IC50 | = | 6 | nM | ALA4308764 | 8.22 | nM | Homo sapiens | ||
6. | ALA4537527 | 14 | Stability | = | 99 | % | ALA4308763 | % | ||||
7. | ALA4537527 | 14 | Stability | = | 85 | % | ALA4308762 | % | ||||
8. | ALA4537527 | 14 | Emax | = | 210 | % | ALA4308761 | % | Homo sapiens | |||
9. | ALA4537527 | 14 | EC50 | = | 56 | nM | ALA4308760 | 7.25 | nM | Homo sapiens | ||
10. | ALA4537527 | 14 | IC50 | = | 110 | nM | ALA4308758 | 6.96 | nM | Homo sapiens | ||
11. | ALA4537527 | 14 | IC50 | = | 4 | nM | ALA4308759 | 8.40 | nM | Homo sapiens |