# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4537786 | 1g | pEC50 | 0 | ALA4350313 | Not Active | Homo sapiens | |||||
2. | ALA4537786 | 1g | FC | 0 | ALA4350322 | Not Active | Homo sapiens | |||||
3. | ALA4537786 | 1g | solubility | > | 0.5 | mM | ALA4350321 | nM | ||||
4. | ALA4537786 | 1g | IC50 | > | 1000 | uM | ALA4350320 | nM | ||||
5. | ALA4537786 | 1g | IC50 | = | 422.4 | uM | ALA4350319 | nM | ||||
6. | ALA4537786 | 1g | INH | = | 25.4 | % | ALA4350303 | % | ||||
7. | ALA4537786 | 1g | Ratio | = | 1.8 | ALA4350315 | ||||||
8. | ALA4537786 | 1g | INH | = | 97.4 | % | ALA4350312 | % | ||||
9. | ALA4537786 | 1g | INH | = | 72.1 | % | ALA4350314 | % | ||||
10. | ALA4537786 | 1g | Activity | = | 6.6 | % | ALA4350311 | % | ||||
11. | ALA4537786 | 1g | Activity | = | 0 | % | ALA4350310 | % | ||||
12. | ALA4537786 | 1g | Activity | = | 25.5 | % | ALA4350309 | % | Homo sapiens | |||
13. | ALA4537786 | 1g | Activity | 0 | ALA4350323 | Active |