# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4537814 | 50d | Papp | = | 25 | 10'-6 cm/s | ALA4429214 | 10'-6 cm/s | ||||
2. | ALA4537814 | 50d | Ratio | = | 1.3 | ALA4429215 | ||||||
3. | ALA4537814 | 50d | Activity | 0 | ALA4429216 | Not Active | Homo sapiens | |||||
4. | ALA4537814 | 50d | Activity | 0 | ALA4429217 | Not Active | Homo sapiens | |||||
5. | ALA4537814 | 50d | EC20 | > | 86 | uM | ALA4429218 | uM | Homo sapiens | |||
6. | ALA4537814 | 50d | Activity | 0 | ALA4429219 | Active | Homo sapiens | |||||
7. | ALA4537814 | 50d | Activity | 0 | ALA4429220 | Active | Homo sapiens | |||||
8. | ALA4537814 | 50d | Activity | 0 | ALA4429221 | Active | Homo sapiens | |||||
9. | ALA4537814 | 50d | Activity | 0 | ALA4429222 | Active | Homo sapiens | |||||
10. | ALA4537814 | 50d | Activity | 0 | ALA4429223 | Active | Homo sapiens | |||||
11. | ALA4537814 | 50d | Fabs | = | 55 | % | ALA4429224 | % | ||||
12. | ALA4537814 | 50d | Tmax | = | 1 | hr | ALA4429225 | hr | ||||
13. | ALA4537814 | 50d | Tmax | = | 0.5 | hr | ALA4429226 | hr | ||||
14. | ALA4537814 | 50d | Cmax | = | 65 | ng/ml | ALA4429227 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
15. | ALA4537814 | 50d | Cmax | = | 1710 | ng/g | ALA4429228 | ng/g | ||||
16. | ALA4537814 | 50d | Ratio | = | 14 | ALA4429229 | ||||||
17. | ALA4537814 | 50d | ERH | = | 0.9 | ALA4429230 | ||||||
18. | ALA4537814 | 50d | Tmax | = | 0.5 | hr | ALA4429231 | hr | ||||
19. | ALA4537814 | 50d | CLH | = | 5 | uL/min | ALA4429232 | uL/min | ||||
20. | ALA4537814 | 50d | CLH | = | 60 | uL/min | ALA4429233 | uL/min |