# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4538610 | 14j | t1/2 | > | 60 | min | ALA5223629 | hr | ||||
2. | ALA4538610 | 14j | CLH | < | 38 | ml/min.kg | ALA5223628 | mL.min-1.kg-1 | ||||
3. | ALA4538610 | 14j | CL | < | 9.6 | microL/min/mg | ALA5223627 | mL.min-1.g-1 | ||||
4. | ALA4538610 | 14j | Activity | > | 200 | % | ALA5223626 | % | Homo sapiens | |||
5. | ALA4538610 | 14j | Activity | > | 60 | % | ALA5223625 | % | Homo sapiens | |||
6. | ALA4538610 | 14j | Activity | > | 150 | % | ALA5223624 | % | Homo sapiens | |||
7. | ALA4538610 | 14j | Activity | = | 60 | % | ALA5223623 | % | Homo sapiens | |||
8. | ALA4538610 | 14j | Activity | = | 70 | % | ALA5223622 | % | Homo sapiens | |||
9. | ALA4538610 | 14j | Activity | = | 6.6 | % | ALA5223621 | % | Homo sapiens | |||
10. | ALA4538610 | 14j | Activity | = | 13 | % | ALA5223620 | % | Homo sapiens | |||
11. | ALA4538610 | 14j | Activity | = | 27 | % | ALA5223619 | % | Homo sapiens | |||
12. | ALA4538610 | 14j | IC50 | = | 3.3 | uM | ALA5223610 | 5.48 | nM | Homo sapiens | ||
13. | ALA4538610 | 14j | IC50 | = | 1 | uM | ALA5223609 | 6.00 | nM | Homo sapiens | ||
14. | ALA4538610 | 14j | IC50 | = | 1 | uM | ALA5223608 | 6.00 | nM | Homo sapiens | ||
15. | ALA4538610 | 14j | IC50 | = | 1 | uM | ALA5223607 | 6.00 | nM | Homo sapiens | ||
16. | ALA4538610 | 14j | IC50 | = | 1 | uM | ALA5223606 | 6.00 | nM | Homo sapiens | ||
17. | ALA4538610 | 14j | Kd | = | 0.37 | uM | ALA5223605 | 6.43 | nM | Homo sapiens | ||
18. | ALA4538610 | 14j | IC50 | = | 0.47 | uM | ALA5223604 | 6.33 | nM | Homo sapiens | ||
19. | ALA4538610 | 14j | Fu | = | 7.6 | % | ALA4380938 | |||||
20. | ALA4538610 | 14j | Activity | 0 | ALA4380928 | Active | Homo sapiens |