# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4539102 | 5e | INH | 0 | ALA4316041 | Active | % | |||||
2. | ALA4539102 | 5e | INH | 0 | ALA4316040 | Not Active | % | |||||
3. | ALA4539102 | 5e | EC50 | = | 0.24 | uM | ALA4316039 | 6.62 | nM | Homo sapiens | ||
4. | ALA4539102 | 5e | EC50 | = | 12.02 | uM | ALA4316038 | 4.92 | nM | Homo sapiens | ||
5. | ALA4539102 | 5e | Activity | 0 | ALA4316038 | Dose-dependent effect | Homo sapiens | |||||
6. | ALA4539102 | 5e | Activity | 0 | ALA4316027 | Not Active | Homo sapiens | |||||
7. | ALA4539102 | 5e | Ratio TD50/ED50 | = | 9.09 | ALA4316037 | Mus musculus | |||||
8. | ALA4539102 | 5e | TD50 | = | 372.39 | mg kg-1 | ALA4316028 | mg kg-1 | ||||
9. | ALA4539102 | 5e | ED50 | = | 40.95 | mg kg-1 | ALA4316036 | mg.kg-1 | Mus musculus | |||
10. | ALA4539102 | 5e | Activity | 0 | ALA4316035 | Active | Mus musculus | |||||
11. | ALA4539102 | 5e | Activity | 0 | ALA4316034 | Active | Mus musculus | |||||
12. | ALA4539102 | 5e | Activity | 0 | ALA4316033 | Active | Mus musculus | |||||
13. | ALA4539102 | 5e | Activity | 0 | ALA4316032 | Not Active | Mus musculus | |||||
14. | ALA4539102 | 5e | IC50 | = | 0.334 | uM | ALA4316029 | 6.48 | nM | Mus musculus |