| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4539521 | 2 | Ratio | = | 0.95 | ALA4399601 | ||||||
| 2. | ALA4539521 | 2 | permeability | = | 20.1 | 10'-6 cm/s | ALA4399581 | 10'-6 cm/s | ||||
| 3. | ALA4539521 | 2 | Vdss | = | 1.22 | L/Kg | ALA4399597 | L.kg-1 | ||||
| 4. | ALA4539521 | 2 | t1/2 | = | 2.5 | hr | ALA4399596 | hr | ||||
| 5. | ALA4539521 | 2 | CL | = | 22 | ml/min.kg | ALA4399595 | mL.min-1.kg-1 | ||||
| 6. | ALA4539521 | 2 | CL free | = | 33 | uL/min | ALA4399594 | uL/min | ||||
| 7. | ALA4539521 | 2 | CL free | = | 24 | uL/min | ALA4399593 | uL/min | ||||
| 8. | ALA4539521 | 2 | logD | = | 2.9 | ALA4399580 | ||||||
| 9. | ALA4539521 | 2 | Ki | = | 86 | nM | ALA4399592 | 7.07 | nM | Homo sapiens | ||
| 10. | ALA4539521 | 2 | Ki | = | 210 | nM | ALA4399589 | 6.68 | nM | Homo sapiens | ||
| 11. | ALA4539521 | 2 | Ki | = | 240 | nM | ALA4399586 | 6.62 | nM | Homo sapiens | ||
| 12. | ALA4539521 | 2 | Ki | = | 465 | nM | ALA4399585 | 6.33 | nM | Homo sapiens | ||
| 13. | ALA4539521 | 2 | Ki | = | 14 | nM | ALA4399584 | 7.85 | nM | Homo sapiens |
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