| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4539831 | 5a27 | INH | = | 90.9 | % | ALA4387890 | % | ||||
| 2. | ALA4539831 | 5a27 | F | = | 26.62 | % | ALA4387897 | % | ||||
| 3. | ALA4539831 | 5a27 | Stability | 0 | ALA4387896 | Stable | % | |||||
| 4. | ALA4539831 | 5a27 | INH | 0 | ALA4387902 | Active | % | Mus musculus | ||||
| 5. | ALA4539831 | 5a27 | INH | 0 | ALA4387901 | Active | % | |||||
| 6. | ALA4539831 | 5a27 | INH | 0 | ALA4387900 | Active | % | |||||
| 7. | ALA4539831 | 5a27 | INH | 0 | ALA4387907 | Active | % | |||||
| 8. | ALA4539831 | 5a27 | AUCt | = | 34.4 | ug/L.hr | ALA4387911 | ng.hr.mL-1 | ||||
| 9. | ALA4539831 | 5a27 | AUCt | = | 231.2 | ug/L.hr | ALA4387910 | ng.hr.mL-1 | ||||
| 10. | ALA4539831 | 5a27 | MRT(t) | = | 11.3 | hr | ALA4387915 | hr | ||||
| 11. | ALA4539831 | 5a27 | MRT(t) | = | 7.8 | hr | ALA4387914 | hr | ||||
| 12. | ALA4539831 | 5a27 | t1/2 | = | 0.2 | hr | ALA4387919 | hr | ||||
| 13. | ALA4539831 | 5a27 | t1/2 | = | 6.7 | hr | ALA4387918 | hr | ||||
| 14. | ALA4539831 | 5a27 | CLz/F | = | 404.4 | L/hr/kg | ALA4387923 | L/hr/kg | ||||
| 15. | ALA4539831 | 5a27 | CLz/F | = | 5062.6 | L/hr/kg | ALA4387922 | L/hr/kg | ||||
| 16. | ALA4539831 | 5a27 | Cmax | = | 16.4 | ug/L | ALA4387927 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 17. | ALA4539831 | 5a27 | Cmax | = | 113.3 | ug/L | ALA4387926 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 18. | ALA4539831 | 5a27 | Activity | 0 | ALA4387929 | Active | Mus musculus | |||||
| 19. | ALA4539831 | 5a27 | Activity | 0 | ALA4387930 | Active | Mus musculus | |||||
| 20. | ALA4539831 | 5a27 | Activity | 0 | ALA4387932 | Active | Mus musculus |
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