# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4542153 | 21b | Activity | 0 | ALA4411953 | Dose-dependent effect | Homo sapiens | |||||
2. | ALA4542153 | 21b | Activity | 0 | ALA4411949 | Not Active | Rattus norvegicus | |||||
3. | ALA4542153 | 21b | Activity | = | 40 | % | ALA4411944 | % | Rattus norvegicus | |||
4. | ALA4542153 | 21b | Activity | = | 40 | % | ALA4411943 | % | Rattus norvegicus | |||
5. | ALA4542153 | 21b | Activity | 0 | ALA4411942 | Dose-dependent effect | Rattus norvegicus | |||||
6. | ALA4542153 | 21b | Activity | 0 | ALA4411941 | Dose-dependent effect | Rattus norvegicus | |||||
7. | ALA4542153 | 21b | Activity | 0 | ALA4411940 | Active | Rattus norvegicus | |||||
8. | ALA4542153 | 21b | Activity | 0 | ALA4411939 | Active | Mus musculus | |||||
9. | ALA4542153 | 21b | CLH | = | 23.77 | ml/min/mg | ALA4411925 | mL.min-1.g-1 | ||||
10. | ALA4542153 | 21b | t1/2 | = | 9.16 | min | ALA4411924 | hr | ||||
11. | ALA4542153 | 21b | Activity | 0 | ALA4411919 | Active | Homo sapiens | |||||
12. | ALA4542153 | 21b | Activity | < | 30 | % | ALA4411918 | % | ||||
13. | ALA4542153 | 21b | Ki | = | 0.326 | uM | ALA4411915 | 6.49 | nM | Homo sapiens | ||
14. | ALA4542153 | 21b | IC50 | = | 0.13 | uM | ALA4411916 | 6.89 | nM | Homo sapiens | ||
15. | ALA4542153 | 21b | Activity | = | 31 | % | ALA4411917 | % | Homo sapiens |