| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4542825 | 9a | Ratio ED50 | = | 19 | ALA4310633 | Rattus norvegicus | |||||
| 2. | ALA4542825 | 9a | Ratio ED50 | = | 266 | ALA4310632 | ||||||
| 3. | ALA4542825 | 9a | ED50 | = | 10.65 | mg kg-1 | ALA4310631 | mg.kg-1 | Rattus norvegicus | |||
| 4. | ALA4542825 | 9a | ED50 | = | 0.57 | mg kg-1 | ALA4310629 | mg.kg-1 | Rattus norvegicus | |||
| 5. | ALA4542825 | 9a | ED50 | = | 0.04 | mg kg-1 | ALA4310627 | mg.kg-1 | Mustela putorius furo | |||
| 6. | ALA4542825 | 9a | Ke | = | 3.8 | nM | ALA4310626 | nM | Homo sapiens | |||
| 7. | ALA4542825 | 9a | Ke | = | 6.2 | nM | ALA4310625 | nM | Homo sapiens | |||
| 8. | ALA4542825 | 9a | Stability | > | 80 | % | ALA4310624 | % | ||||
| 9. | ALA4542825 | 9a | Stability | 0 | ALA4310623 | Stable | % | |||||
| 10. | ALA4542825 | 9a | Cmax | 0 | ALA4310621 | Not Determined | ||||||
| 11. | ALA4542825 | 9a | F | = | 50 | % | ALA4310619 | % | ||||
| 12. | ALA4542825 | 9a | CL | = | 41 | ml/min.kg | ALA4310618 | mL.min-1.kg-1 | ||||
| 13. | ALA4542825 | 9a | Stability | = | 88 | % | ALA4310617 | % | ||||
| 14. | ALA4542825 | 9a | Stability | = | 95 | % | ALA4310616 | % | ||||
| 15. | ALA4542825 | 9a | Ki | = | 2 | nM | ALA4310615 | 8.70 | nM | Homo sapiens | ||
| 16. | ALA4542825 | 9a | Ki | = | 3.4 | nM | ALA4310614 | 8.47 | nM | Homo sapiens |
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