# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4545886 | 34 | F | = | 96 | % | ALA4355767 | % | ||||
2. | ALA4545886 | 34 | Vdss | = | 2.88 | L/Kg | ALA4355764 | L.kg-1 | ||||
3. | ALA4545886 | 34 | t1/2 | = | 1.63 | hr | ALA4355762 | hr | ||||
4. | ALA4545886 | 34 | CL | = | 53.6 | ml/min.kg | ALA4355760 | mL.min-1.kg-1 | ||||
5. | ALA4545886 | 34 | AUC/dose | = | 1.15 | uM.hr.kg/mg | ALA4355758 | uM.hr.kg/mg | ||||
6. | ALA4545886 | 34 | EC50 | = | 28 | nM | ALA4355755 | 7.55 | nM | Rattus norvegicus | ||
7. | ALA4545886 | 34 | Ki | = | 3.3 | nM | ALA4355754 | 8.48 | nM | Homo sapiens | ||
8. | ALA4545886 | 34 | Ki | > | 10000 | nM | ALA4355756 | nM | Homo sapiens |