# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4548488 | Ex 126 | T/C | = | 0.44 | ALA4421198 | ||||||
2. | ALA4548488 | Ex 126 | T/C | = | 0.46 | ALA4421196 | Homo sapiens | |||||
3. | ALA4548488 | Ex 126 | F | = | 33 | % | ALA4421193 | % | ||||
4. | ALA4548488 | Ex 126 | F | = | 67 | % | ALA4421192 | % | ||||
5. | ALA4548488 | Ex 126 | t1/2 | = | 1.8 | hr | ALA4421191 | hr | ||||
6. | ALA4548488 | Ex 126 | t1/2 | = | 2.3 | hr | ALA4421190 | hr | ||||
7. | ALA4548488 | Ex 126 | Cmax | = | 35 | uM | ALA4421189 | nM | ||||
8. | ALA4548488 | Ex 126 | Cmax | = | 100 | uM | ALA4421188 | nM | ||||
9. | ALA4548488 | Ex 126 | AUC | = | 106 | uM.hr | ALA4421187 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
10. | ALA4548488 | Ex 126 | AUC | = | 413 | uM.hr | ALA4421186 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
11. | ALA4548488 | Ex 126 | IC50 | > | 100 | uM | ALA4421185 | nM | Sus scrofa | |||
12. | ALA4548488 | Ex 126 | IC50 | > | 100 | uM | ALA4421184 | nM | Homo sapiens | |||
13. | ALA4548488 | Ex 126 | IC50 | > | 100 | uM | ALA4421183 | nM | Homo sapiens | |||
14. | ALA4548488 | Ex 126 | IC50 | = | 0.24 | uM | ALA4421181 | 6.62 | nM | Homo sapiens | ||
15. | ALA4548488 | Ex 126 | IC50 | = | 0.7 | uM | ALA4421179 | 6.16 | nM | |||
16. | ALA4548488 | Ex 126 | IC50 | > | 100 | uM | ALA4421175 | nM |