# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4549976 | 17 | t1/2 | = | 3.6 | hr | ALA4339130 | hr | ||||
2. | ALA4549976 | 17 | AUC | = | 30 | uM.hr | ALA4339129 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
3. | ALA4549976 | 17 | Cmax | = | 3.3 | uM | ALA4339128 | nM | ||||
4. | ALA4549976 | 17 | IC50 | > | 10 | uM | ALA4339127 | nM | Homo sapiens | |||
5. | ALA4549976 | 17 | IC50 | > | 10 | uM | ALA4339126 | nM | Homo sapiens | |||
6. | ALA4549976 | 17 | IC50 | > | 10 | uM | ALA4339125 | nM | Homo sapiens | |||
7. | ALA4549976 | 17 | IC50 | > | 10 | uM | ALA4339124 | nM | Homo sapiens | |||
8. | ALA4549976 | 17 | IC50 | = | 320 | nM | ALA4339120 | 6.50 | nM | Homo sapiens | ||
9. | ALA4549976 | 17 | IC50 | > | 10000 | nM | ALA4339118 | nM | Homo sapiens | |||
10. | ALA4549976 | 17 | Drug metabolism | = | 16 | % | ALA4339117 | % | ||||
11. | ALA4549976 | 17 | t1/2 | > | 180 | min | ALA4339116 | hr | Homo sapiens | |||
12. | ALA4549976 | 17 | t1/2 | = | 165 | min | ALA4339115 | hr | ||||
13. | ALA4549976 | 17 | t1/2 | > | 180 | min | ALA4339114 | hr | ||||
14. | ALA4549976 | 17 | IC50 | = | 21 | nM | ALA4339113 | 7.68 | nM | Homo sapiens | ||
15. | ALA4549976 | 17 | IC50 | = | 93 | nM | ALA4339112 | 7.03 | nM | Homo sapiens |