# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4550982 | 10ab | INH | 0 | ALA4366987 | Active | % | Bos taurus | ||||
2. | ALA4550982 | 10ab | Ratio IC50 | = | 1.8 | ALA4367028 | ||||||
3. | ALA4550982 | 10ab | IC50 | = | 25.2 | nM | ALA4367027 | 7.60 | nM | |||
4. | ALA4550982 | 10ab | IC50 | = | 13.8 | nM | ALA4367026 | 7.86 | nM | Homo sapiens | ||
5. | ALA4550982 | 10ab | Ratio IC50 | = | 0.8 | ALA4367025 | ||||||
6. | ALA4550982 | 10ab | IC50 | = | 3.9 | nM | ALA4367024 | 8.41 | nM | |||
7. | ALA4550982 | 10ab | IC50 | = | 5.2 | nM | ALA4367023 | 8.28 | nM | Homo sapiens | ||
8. | ALA4550982 | 10ab | CLH | = | 3.1 | ml/min.kg | ALA4366999 | mL.min-1.kg-1 | ||||
9. | ALA4550982 | 10ab | t1/2 | = | 6.7 | hr | ALA4366998 | hr | ||||
10. | ALA4550982 | 10ab | CLH | = | 25.98 | ml/min.kg | ALA4366997 | mL.min-1.kg-1 | ||||
11. | ALA4550982 | 10ab | t1/2 | = | 1.8 | hr | ALA4366996 | hr | ||||
12. | ALA4550982 | 10ab | CLH | = | 23.6 | ml/min.kg | ALA4366995 | mL.min-1.kg-1 | ||||
13. | ALA4550982 | 10ab | t1/2 | = | 2.42 | hr | ALA4366994 | hr | ||||
14. | ALA4550982 | 10ab | Activity | = | 35.6 | % | ALA4366993 | % | Homo sapiens | |||
15. | ALA4550982 | 10ab | Activity | = | 25.9 | % | ALA4366992 | % | Homo sapiens | |||
16. | ALA4550982 | 10ab | Activity | = | 48.5 | % | ALA4366991 | % | Homo sapiens | |||
17. | ALA4550982 | 10ab | INH | = | 59 | % | ALA4366990 | % | Homo sapiens | |||
18. | ALA4550982 | 10ab | Activity | 0 | ALA4366989 | Active | Homo sapiens | |||||
19. | ALA4550982 | 10ab | Activity | 0 | ALA4366988 | Active | Homo sapiens | |||||
20. | ALA4550982 | 10ab | IC50 | = | 3.2 | nM | ALA4366986 | 8.49 | nM | Homo sapiens |