# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4552641 | 14 | t1/2 | = | 51 | min | ALA4400659 | hr | ||||
2. | ALA4552641 | 14 | INH | = | 21 | % | ALA4400656 | % | Homo sapiens | |||
3. | ALA4552641 | 14 | INH | = | 28 | % | ALA4400655 | % | Homo sapiens | |||
4. | ALA4552641 | 14 | Selectivity Index | = | 11000 | ALA4400650 | ||||||
5. | ALA4552641 | 14 | Activity | < | 20 | % | ALA4400649 | % | Homo sapiens | |||
6. | ALA4552641 | 14 | INH | = | 30 | % | ALA4400646 | % | Mus musculus | |||
7. | ALA4552641 | 14 | IC50 | = | 11.6 | nM | ALA4400644 | 7.94 | nM | Mus musculus | ||
8. | ALA4552641 | 14 | Ratio IC50 | = | 3.4 | ALA4400643 | ||||||
9. | ALA4552641 | 14 | IC50 | = | 4.8 | nM | ALA4400642 | 8.32 | nM | Homo sapiens | ||
10. | ALA4552641 | 14 | IC50 | = | 1.4 | nM | ALA4400641 | 8.85 | nM | Homo sapiens |