# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4555799 | 20a | IC50 | > | 200 | nM | ALA4403344 | nM | Homo sapiens | |||
2. | ALA4555799 | 20a | IC50 | > | 200 | nM | ALA4403340 | nM | Homo sapiens | |||
3. | ALA4555799 | 20a | IC50 | < | 20 | nM | ALA4403338 | nM | Homo sapiens | |||
4. | ALA4555799 | 20a | IC50 | 0 | ALA4742488 | Not Determined | Homo sapiens | |||||
5. | ALA4555799 | 20a | IC50 | <= | 20 | nM | ALA4742487 | nM | Homo sapiens | |||
6. | ALA4555799 | 20a | IC50 | = | 0.2 | uM | ALA4742486 | 6.70 | nM | Homo sapiens | ||
7. | ALA4555799 | 20a | IC50 | = | 0.2 | uM | ALA4742485 | 6.70 | nM | Homo sapiens | ||
8. | ALA4555799 | 20a | IC50 | = | 0.2 | uM | ALA4742484 | 6.70 | nM | Homo sapiens | ||
9. | ALA4555799 | 20a | IC50 | < | 20 | nM | ALA4742483 | nM | Homo sapiens | |||
10. | ALA4555799 | 20a | K | = | 0.004 | /s | ALA5043167 | /s | Homo sapiens | |||
11. | ALA4555799 | 20a | IC50 | = | 29 | nM | ALA5043166 | 7.54 | nM | Homo sapiens | ||
12. | ALA4555799 | 20a | IC50 | = | 23 | nM | ALA5043165 | 7.64 | nM | Homo sapiens | ||
13. | ALA4555799 | 20a | Kd | = | 0.33 | nM | ALA5043164 | 9.48 | nM | Homo sapiens | ||
14. | ALA4555799 | 20a | EC50 | = | 40 | nM | ALA5043163 | 7.40 | nM | Homo sapiens | ||
15. | ALA4555799 | 20a | IC50 | = | 102 | nM | ALA5043162 | 6.99 | nM | Homo sapiens | ||
16. | ALA4555799 | 20a | logD | = | 1.78 | ALA5043160 | ||||||
17. | ALA4555799 | 20a | CLH | = | 109 | ml/min.kg | ALA5043159 | mL.min-1.kg-1 | ||||
18. | ALA4555799 | 20a | Papp | = | 5.26 | 10^-6 cm/s | ALA5043158 | 10^-6 cm/s | ||||
19. | ALA4555799 | 20a | CL free | = | 457 | ml/min.kg | ALA5043157 | mL.min-1.kg-1 | ||||
20. | ALA4555799 | 20a | F | = | 39 | % | ALA5043156 | % |