# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | GSK2603566A | 39 | permeability | = | 80 | nm/s | ALA4355843 | nm/s | ||||
2. | GSK2603566A | 39 | F | = | 98 | % | ALA4355842 | % | ||||
3. | GSK2603566A | 39 | t1/2 | = | 1.8 | hr | ALA4355841 | hr | ||||
4. | GSK2603566A | 39 | Vdss | = | 0.5 | L/Kg | ALA4355840 | L.kg-1 | ||||
5. | GSK2603566A | 39 | CL | = | 8 | ml/min.Kg | ALA4355839 | mL.min-1.kg-1 | ||||
6. | GSK2603566A | 39 | pIC50 | = | 7.4 | ALA4355838 | 7.40 | nM | ||||
7. | GSK2603566A | 39 | pIC50 | = | 8.4 | ALA4355837 | 8.40 | nM | ||||
8. | GSK2603566A | 39 | pIC50 | = | 8.4 | ALA4355836 | 8.40 | nM | Homo sapiens | |||
9. | GSK2603566A | 39 | pIC50 | = | 7.8 | ALA4355835 | 7.80 | nM | Homo sapiens |