# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4558456 | 30 | F | = | 7 | % | ALA4367205 | % | ||||
2. | ALA4558456 | 30 | AUC | = | 23.2 | hr.ng/ml | ALA4367204 | ng.hr.mL-1 | ||||
3. | ALA4558456 | 30 | beta t1/2 | = | 2.1 | hr | ALA4367203 | hr | ||||
4. | ALA4558456 | 30 | Vdss | = | 13.4 | L/Kg | ALA4367202 | L.kg-1 | ||||
5. | ALA4558456 | 30 | CLH | = | 114.6 | ml/min.kg | ALA4367201 | mL.min-1.kg-1 | ||||
6. | ALA4558456 | 30 | Stability | = | 19 | % | ALA4367200 | % | ||||
7. | ALA4558456 | 30 | Stability | = | 74 | % | ALA4367199 | % | ||||
8. | ALA4558456 | 30 | IC50 | > | 10 | uM | ALA4367198 | nM | Homo sapiens | |||
9. | ALA4558456 | 30 | IC50 | > | 10 | uM | ALA4367197 | nM | Homo sapiens | |||
10. | ALA4558456 | 30 | IC50 | > | 10 | uM | ALA4367196 | nM | Homo sapiens | |||
11. | ALA4558456 | 30 | IC50 | > | 10 | uM | ALA4367195 | nM | Homo sapiens | |||
12. | ALA4558456 | 30 | IC50 | > | 10 | uM | ALA4367194 | nM | Homo sapiens | |||
13. | ALA4558456 | 30 | IC50 | = | 58 | nM | ALA4367190 | 7.24 | nM | Homo sapiens | ||
14. | ALA4558456 | 30 | IC50 | = | 27 | nM | ALA4367191 | 7.57 | nM | Homo sapiens |