# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | YQ128 | 17; YQ128 | Activity | = | 99 | % | ALA5140068 | % | Homo sapiens | |||
2. | YQ128 | 17; YQ128 | Activity | = | 106 | % | ALA5140067 | % | Mus musculus | |||
3. | YQ128 | 17; YQ128 | IC50 | = | 0.3 | uM | ALA5140066 | 6.52 | nM | Mus musculus | ||
4. | YQ128 | 17; YQ128 | F | = | 10 | % | ALA4416633 | % | ||||
5. | YQ128 | 17; YQ128 | Cmax | = | 73 | ng/ml | ALA4416632 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
6. | YQ128 | 17; YQ128 | Tmax | = | 12 | hr | ALA4416631 | hr | ||||
7. | YQ128 | 17; YQ128 | beta t1/2 | = | 6.6 | hr | ALA4416630 | hr | ||||
8. | YQ128 | 17; YQ128 | CL | = | 41 | ml/min.kg | ALA4416629 | mL.min-1.kg-1 | ||||
9. | YQ128 | 17; YQ128 | Vdss | = | 8.5 | L/Kg | ALA4416628 | L.kg-1 | ||||
10. | YQ128 | 17; YQ128 | Ratio | = | 25 | ALA4416627 | ||||||
11. | YQ128 | 17; YQ128 | BPR | = | 0.82 | ALA4416626 | ||||||
12. | YQ128 | 17; YQ128 | BPR | = | 0.36 | ALA4416625 | ||||||
13. | YQ128 | 17; YQ128 | BPR | = | 0.077 | ALA4416624 | ||||||
14. | YQ128 | 17; YQ128 | Cp | = | 8 | ng/ml | ALA4416623 | ng/ml | ||||
15. | YQ128 | 17; YQ128 | Cp | = | 57.6 | ng/ml | ALA4416622 | ng/ml | ||||
16. | YQ128 | 17; YQ128 | Cp | = | 277.33 | ng/ml | ALA4416621 | ng/ml | ||||
17. | YQ128 | 17; YQ128 | Drug uptake | = | 6.58 | ng/g | ALA4416620 | ng/g | ||||
18. | YQ128 | 17; YQ128 | Drug uptake | = | 20.48 | ng/g | ALA4416619 | ng/g | ||||
19. | YQ128 | 17; YQ128 | Drug uptake | = | 21.25 | ng/g | ALA4416618 | ng/g | ||||
20. | YQ128 | 17; YQ128 | Ratio | = | 0.22 | ALA4416617 |