# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4564074 | 7e | Papp | 0 | ALA4403255 | Not Determined | ||||||
2. | ALA4564074 | 7e | Papp | 0 | ALA4403254 | Not Determined | ||||||
3. | ALA4564074 | 7e | F | 0 | ALA4403249 | Not Determined | % | |||||
4. | ALA4564074 | 7e | t1/2 | = | 0.6 | hr | ALA4403248 | hr | ||||
5. | ALA4564074 | 7e | AUC | = | 9.97 | uM.hr | ALA4403247 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
6. | ALA4564074 | 7e | Cmax | = | 10.16 | uM | ALA4403246 | nM | ||||
7. | ALA4564074 | 7e | Stability | = | 70 | % | ALA4403244 | % | ||||
8. | ALA4564074 | 7e | IC50 | = | 36 | uM | ALA4403243 | 4.44 | nM | Homo sapiens | ||
9. | ALA4564074 | 7e | IC50 | = | 3.6 | uM | ALA4403242 | 5.44 | nM | Homo sapiens | ||
10. | ALA4564074 | 7e | IC50 | > | 100 | uM | ALA4403241 | nM | Sus scrofa | |||
11. | ALA4564074 | 7e | IC50 | = | 46.2 | uM | ALA4403240 | 4.33 | nM | Homo sapiens | ||
12. | ALA4564074 | 7e | IC50 | = | 29.2 | uM | ALA4403239 | 4.54 | nM | Homo sapiens | ||
13. | ALA4564074 | 7e | Ratio IC50 | >= | 10 | ALA4403238 | ||||||
14. | ALA4564074 | 7e | IC50 | = | 6.78 | uM | ALA4403237 | 5.17 | nM | Homo sapiens | ||
15. | ALA4564074 | 7e | IC50 | = | 6.91 | uM | ALA4403236 | 5.16 | nM | |||
16. | ALA4564074 | 7e | IC50 | = | 0.38 | uM | ALA4403232 | 6.42 | nM | Homo sapiens |