| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4564517 | 9g | Activity | < | 5 | % | ALA4421202 | % | ||||
| 2. | ALA4564517 | 9g | T/C | = | 0.56 | ALA4421195 | Homo sapiens | |||||
| 3. | ALA4564517 | 9g | F | = | 39 | % | ALA4421192 | % | ||||
| 4. | ALA4564517 | 9g | t1/2 | = | 1.3 | hr | ALA4421190 | hr | ||||
| 5. | ALA4564517 | 9g | Cmax | = | 6.7 | uM | ALA4421188 | nM | ||||
| 6. | ALA4564517 | 9g | AUC | = | 11 | uM.hr | ALA4421186 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 7. | ALA4564517 | 9g | IC50 | > | 100 | uM | ALA4421185 | nM | Sus scrofa | |||
| 8. | ALA4564517 | 9g | IC50 | = | 87 | uM | ALA4421184 | 4.06 | nM | Homo sapiens | ||
| 9. | ALA4564517 | 9g | IC50 | > | 100 | uM | ALA4421183 | nM | Homo sapiens | |||
| 10. | ALA4564517 | 9g | IC50 | = | 0.19 | uM | ALA4421182 | 6.72 | nM | Homo sapiens | ||
| 11. | ALA4564517 | 9g | IC50 | = | 2 | uM | ALA4421180 | 5.70 | nM | Homo sapiens | ||
| 12. | ALA4564517 | 9g | IC50 | = | 1.1 | uM | ALA4421178 | 5.96 | nM | |||
| 13. | ALA4564517 | 9g | IC50 | > | 100 | uM | ALA4421175 | nM | ||||
| 14. | ALA4564517 | 9g | Papp | = | 17 | 10'-6 cm/s | ALA4305238 | 10'-6 cm/s | ||||
| 15. | ALA4564517 | 9g | Papp | = | 8 | 10'-6 cm/s | ALA4305237 | 10'-6 cm/s | ||||
| 16. | ALA4564517 | 9g | IC50 | = | 4.6 | uM | ALA4305236 | 5.34 | nM | Homo sapiens | ||
| 17. | ALA4564517 | 9g | IC50 | = | 87 | uM | ALA4305234 | 4.06 | nM | Homo sapiens | ||
| 18. | ALA4564517 | 9g | IC50 | > | 100 | uM | ALA4305233 | nM | Homo sapiens | |||
| 19. | ALA4564517 | 9g | IC50 | = | 49 | uM | ALA4305232 | 4.31 | nM | Homo sapiens | ||
| 20. | ALA4564517 | 9g | Stability | = | 60 | % | ALA4305224 | % |
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