| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4564973 | 50 | F | = | 12 | % | ALA4390039 | % | ||||
| 2. | ALA4564973 | 50 | AUC | = | 1889 | hr.ng/ml | ALA4390038 | ng.hr.mL-1 | ||||
| 3. | ALA4564973 | 50 | beta t1/2 | = | 2.5 | hr | ALA4390037 | hr | ||||
| 4. | ALA4564973 | 50 | Vdss | = | 0.21 | L/Kg | ALA4390036 | L.kg-1 | ||||
| 5. | ALA4564973 | 50 | CL | = | 11 | % | ALA4389075 | % | ||||
| 6. | ALA4564973 | 50 | CL | = | 6.2 | ml/min.kg | ALA4390035 | mL.min-1.kg-1 | ||||
| 7. | ALA4564973 | 50 | Fu | = | 0.13 | % | ALA4390034 | |||||
| 8. | ALA4564973 | 50 | Fu | = | 1 | % | ALA4390033 | |||||
| 9. | ALA4564973 | 50 | CLH | = | 10 | % | ALA4390032 | % | ||||
| 10. | ALA4564973 | 50 | CLH | = | 53 | % | ALA4389076 | % | ||||
| 11. | ALA4564973 | 50 | Ratio | = | 11 | ALA4390031 | ||||||
| 12. | ALA4564973 | 50 | Papp | = | 4 | 10'-6 cm/s | ALA4390030 | 10'-6 cm/s | ||||
| 13. | ALA4564973 | 50 | Kinetic_solubility | = | 94 | ug ml-1 | ALA4390029 | ug.mL-1 | ||||
| 14. | ALA4564973 | 50 | Kinetic_solubility | = | 8 | ug ml-1 | ALA4390028 | ug.mL-1 | ||||
| 15. | ALA4564973 | 50 | logD | = | 2.6 | ALA4390027 | ||||||
| 16. | ALA4564973 | 50 | IC50 | = | 92 | nM | ALA4390026 | 7.04 | nM | Homo sapiens | ||
| 17. | ALA4564973 | 50 | IC50 | = | 251 | nM | ALA4390025 | 6.60 | nM | Homo sapiens | ||
| 18. | ALA4564973 | 50 | IC50 | = | 0.238 | uM | ALA4390024 | 6.62 | nM | Homo sapiens | ||
| 19. | ALA4564973 | 50 | INH | = | 80 | % | ALA4390023 | % | Homo sapiens | |||
| 20. | ALA4564973 | 50 | INH | = | 100 | % | ALA4390022 | % | Homo sapiens |
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