| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  PF-05221304 | 38 | IC50 | = | 0.03 | uM | ALA4344284 | 7.52 | nM | Homo sapiens | ||
| 2. | PF-05221304 | 38 | IC50 | = | 0.031 | uM | ALA4344283 | 7.51 | nM | Homo sapiens | ||
| 3. | PF-05221304 | 38 | pIC50 | = | 7.5 | ALA4669981 | 7.50 | nM | Homo sapiens | |||
| 4. | PF-05221304 | 38 | IC50 | = | 0.033 | uM | ALA4669981 | 7.48 | nM | Homo sapiens | ||
| 5. | PF-05221304 | 38 | pIC50 | = | 7.6 | ALA4669980 | 7.60 | nM | Homo sapiens | |||
| 6. | PF-05221304 | 38 | IC50 | = | 0.026 | uM | ALA4669980 | 7.58 | nM | Homo sapiens | ||
| 7. | PF-05221304 | 38 | Papp | = | 14 | 10^-6 cm/s | ALA4669979 | 10^-6 cm/s | ||||
| 8. | PF-05221304 | 38 | logD | = | 1.1 | ALA4669978 | ||||||
| 9. | PF-05221304 | 38 | CLH | < | 3 | uL/min | ALA4669977 | uL/min | ||||
| 10. | PF-05221304 | 38 | Ratio | = | 3.5 | ALA4669974 | Homo sapiens | |||||
| 11. | PF-05221304 | 38 | Ratio | = | 2.5 | ALA4669973 | Homo sapiens | |||||
| 12. | PF-05221304 | 38 | Fu | = | 0.039 | ALA4669972 | ||||||
| 13. | PF-05221304 | 38 | Fu | = | 0.01 | ALA4669971 | ||||||
| 14. | PF-05221304 | 38 | Fu | = | 0.15 | ALA4669970 | ||||||
| 15. | PF-05221304 | 38 | Fu | = | 0.066 | ALA4669969 | ||||||
| 16. | PF-05221304 | 38 | Cp | = | 314 | ng/ml | ALA4669966 | ng/ml | ||||
| 17. | PF-05221304 | 38 | Kp | = | 78 | ALA4669963 | ||||||
| 18. | PF-05221304 | 38 | Drug uptake | = | 24600 | ng/ml | ALA4669960 | ng/ml | ||||
| 19. | PF-05221304 | 38 | Ratio | = | 132 | ALA4669956 | ||||||
| 20. | PF-05221304 | 38 | CL | = | 16 | ml/min.kg | ALA4669954 | mL.min-1.kg-1 |
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