# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4569703 | 2 | IC50 | = | 0.06 | uM | ALA4330597 | 7.22 | nM | Trypanosoma brucei | ||
2. | ALA4569703 | 2 | IC50 | = | 0.45 | uM | ALA4330598 | 6.35 | nM | Homo sapiens | ||
3. | ALA4569703 | 2 | Ratio IC50 | = | 7.5 | ALA4330599 | ||||||
4. | ALA4569703 | 2 | Drug uptake | 0 | ALA4330624 | Active | ||||||
5. | ALA4569703 | 2 | Activity | 0 | ALA4330622 | Active | ||||||
6. | ALA4569703 | 2 | Drug uptake | 0 | ALA4330620 | Active | ||||||
7. | ALA4569703 | 2 | Drug uptake | 0 | ALA4330619 | Tde | ||||||
8. | ALA4569703 | 2 | Drug uptake | = | 36 | % | ALA4330618 | % | ||||
9. | ALA4569703 | 2 | Ka | = | 1.2 | 10'6/M | ALA4330617 | 10'6/M | ||||
10. | ALA4569703 | 2 | Ka | = | 9.2 | 10'5/M | ALA4330616 | 10'5/M | Homo sapiens | |||
11. | ALA4569703 | 2 | Drug uptake | 0 | ALA4330615 | Active | ||||||
12. | ALA4569703 | 2 | Activity | = | 10 | nm | ALA4330613 | nm | Homo sapiens | |||
13. | ALA4569703 | 2 | Activity | 0 | ALA4330612 | Active | ||||||
14. | ALA4569703 | 2 | Activity | 0 | ALA4330611 | Active | ||||||
15. | ALA4569703 | 2 | Activity | 0 | ALA4330610 | Not Active | ||||||
16. | ALA4569703 | 2 | Activity | 0 | ALA4330606 | Active | ||||||
17. | ALA4569703 | 2 | Activity | 0 | ALA4330605 | Active | ||||||
18. | ALA4569703 | 2 | Activity | 0 | ALA4330604 | Non-Toxic | ||||||
19. | ALA4569703 | 2 | Selectivity Index | = | 3 | ALA4330603 | ||||||
20. | ALA4569703 | 2 | TC50 | = | 2.18 | uM | ALA4330602 | uM | Homo sapiens |