# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4570783 | 2 | INH | 0 | ALA4422440 | Active | % | Homo sapiens | ||||
2. | ALA4570783 | 2 | INH | 0 | ALA4422439 | Active | % | Homo sapiens | ||||
3. | ALA4570783 | 2 | CLH | < | 0.02 | ml/min/mg | ALA4422481 | mL.min-1.g-1 | ||||
4. | ALA4570783 | 2 | t1/2 | > | 60 | min | ALA4422480 | hr | ||||
5. | ALA4570783 | 2 | Stability | = | 74 | % | ALA4422479 | % | ||||
6. | ALA4570783 | 2 | Stability | = | 83 | % | ALA4422478 | % | ||||
7. | ALA4570783 | 2 | Stability | = | 91 | % | ALA4422477 | % | ||||
8. | ALA4570783 | 2 | Stability | = | 119 | % | ALA4422476 | % | ||||
9. | ALA4570783 | 2 | Stability | = | 100 | % | ALA4422475 | % | ||||
10. | ALA4570783 | 2 | CLH | = | 0.1 | ml/min/mg | ALA4422474 | mL.min-1.g-1 | ||||
11. | ALA4570783 | 2 | t1/2 | = | 13.5 | min | ALA4422473 | hr | ||||
12. | ALA4570783 | 2 | Stability | = | 21 | % | ALA4422472 | % | ||||
13. | ALA4570783 | 2 | Stability | = | 26 | % | ALA4422471 | % | ||||
14. | ALA4570783 | 2 | Stability | = | 32 | % | ALA4422470 | % | ||||
15. | ALA4570783 | 2 | Stability | = | 45 | % | ALA4422469 | % | ||||
16. | ALA4570783 | 2 | Stability | = | 100 | % | ALA4422468 | % | ||||
17. | ALA4570783 | 2 | IC50 | = | 0.4 | uM | ALA4422457 | 6.40 | nM | Homo sapiens | ||
18. | ALA4570783 | 2 | IC50 | = | 0.4 | uM | ALA4422456 | 6.40 | nM | Homo sapiens |