| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4571380 | 15; MRS7591 | Ki | = | 17.8 | nM | ALA5155979 | 7.75 | nM | Mus musculus | ||
| 2. | ALA4571380 | 15; MRS7591 | Ki | = | 590 | nM | ALA5155978 | 6.23 | nM | Mus musculus | ||
| 3. | ALA4571380 | 15; MRS7591 | t1/2 | = | 16.3 | min | ALA5155976 | hr | ||||
| 4. | ALA4571380 | 15; MRS7591 | t1/2 | = | 15.7 | min | ALA5155975 | hr | ||||
| 5. | ALA4571380 | 15; MRS7591 | t1/2 | = | 7.92 | min | ALA5155974 | hr | ||||
| 6. | ALA4571380 | 15; MRS7591 | Ratio | = | 7.17 | ALA5155973 | ||||||
| 7. | ALA4571380 | 15; MRS7591 | Papp | = | 2.71 | 10^-6 cm/s | ALA5155972 | 10^-6 cm/s | ||||
| 8. | ALA4571380 | 15; MRS7591 | Stability | = | 100 | % | ALA5155971 | % | ||||
| 9. | ALA4571380 | 15; MRS7591 | Stability | = | 84.6 | % | ALA5155970 | % | ||||
| 10. | ALA4571380 | 15; MRS7591 | Stability | = | 91.8 | % | ALA5155969 | % | ||||
| 11. | ALA4571380 | 15; MRS7591 | IC50 | = | 2.23 | uM | ALA5155968 | 5.65 | nM | Homo sapiens | ||
| 12. | ALA4571380 | 15; MRS7591 | IC50 | > | 30 | uM | ALA5155967 | nM | Homo sapiens | |||
| 13. | ALA4571380 | 15; MRS7591 | IC50 | > | 30 | uM | ALA5155966 | nM | Homo sapiens | |||
| 14. | ALA4571380 | 15; MRS7591 | IC50 | = | 14.4 | uM | ALA5155965 | 4.84 | nM | Homo sapiens | ||
| 15. | ALA4571380 | 15; MRS7591 | IC50 | = | 2.89 | uM | ALA5155964 | 5.54 | nM | Homo sapiens | ||
| 16. | ALA4571380 | 15; MRS7591 | Stability | = | 100 | % | ALA5155963 | % | ||||
| 17. | ALA4571380 | 15; MRS7591 | Stability | = | 73.6 | % | ALA5155962 | % | ||||
| 18. | ALA4571380 | 15; MRS7591 | Ki | = | 10.9 | nM | ALA5155957 | 7.96 | nM | Homo sapiens | ||
| 19. | ALA4571380 | 15; MRS7591 | INH | = | 39 | % | ALA5155953 | % | Homo sapiens | |||
| 20. | ALA4571380 | 15; MRS7591 | INH | = | 33 | % | ALA5155951 | % | Homo sapiens |
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