# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4572863 | 6b | CL free | = | 6.1 | L/hr/kg | ALA4428721 | mL.min-1.kg-1 | ||||
2. | ALA4572863 | 6b | CL | = | 0.2 | L/hr/kg | ALA4428720 | mL.min-1.kg-1 | ||||
3. | ALA4572863 | 6b | Activity | = | 5 | % | ALA4428719 | % | Homo sapiens | |||
4. | ALA4572863 | 6b | Activity | = | -1 | % | ALA4428718 | % | Homo sapiens | |||
5. | ALA4572863 | 6b | IC50 | > | 27 | uM | ALA4428717 | nM | Homo sapiens | |||
6. | ALA4572863 | 6b | IC50 | > | 27 | uM | ALA4428716 | nM | Homo sapiens | |||
7. | ALA4572863 | 6b | CLH | < | 14 | uL/min.mg | ALA4428715 | mL.min-1.g-1 | ||||
8. | ALA4572863 | 6b | CLH | < | 14 | uL/min.mg | ALA4428714 | mL.min-1.g-1 | ||||
9. | ALA4572863 | 6b | IC50 | = | 0.5 | nM | ALA4428713 | 9.30 | nM | Mus musculus | ||
10. | ALA4572863 | 6b | IC50 | = | 1.6 | nM | ALA4428712 | 8.80 | nM | Homo sapiens | ||
11. | ALA4572863 | 6b | IC50 | = | 5360 | nM | ALA4428711 | 5.27 | nM | Homo sapiens | ||
12. | ALA4572863 | 6b | IC50 | = | 11000 | nM | ALA4428710 | 4.96 | nM | Homo sapiens | ||
13. | ALA4572863 | 6b | IC50 | = | 3.6 | nM | ALA4428708 | 8.44 | nM | Homo sapiens | ||
14. | ALA4572863 | 6b | IC50 | = | 16800 | nM | ALA4428709 | 4.78 | nM | Homo sapiens |