# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4575590 | 30 | CLH | = | 732 | uL/min | ALA4478463 | uL/min | ||||
2. | ALA4575590 | 30 | CLH | < | 0.1 | uL/min | ALA4478462 | uL/min | ||||
3. | ALA4575590 | 30 | CLH | = | 355 | uL/min | ALA4478461 | uL/min | ||||
4. | ALA4575590 | 30 | CLH | < | 0.1 | uL/min | ALA4478460 | uL/min | ||||
5. | ALA4575590 | 30 | PPB | = | 83.9 | % | ALA4478459 | % | ||||
6. | ALA4575590 | 30 | PPB | = | 99.1 | % | ALA4478458 | % | ||||
7. | ALA4575590 | 30 | t1/2 | > | 24 | hr | ALA4478457 | hr | ||||
8. | ALA4575590 | 30 | t1/2 | > | 24 | hr | ALA4478456 | hr | ||||
9. | ALA4575590 | 30 | t1/2 | > | 24 | hr | ALA4478455 | hr | ||||
10. | ALA4575590 | 30 | solubility | = | 1091 | uM | ALA4478454 | nM | ||||
11. | ALA4575590 | 30 | IC50 | = | 0.042 | uM | ALA4478453 | 7.38 | nM | Human immunodeficiency virus 1 | ||
12. | ALA4575590 | 30 | EC50 | = | 0.3 | uM | ALA4478448 | 6.52 | nM | Human immunodeficiency virus 1 | ||
13. | ALA4575590 | 30 | Ratio CC50/EC50 | = | 380 | ALA4478447 | ||||||
14. | ALA4575590 | 30 | CC50 | = | 23 | uM | ALA4478446 | nM | Homo sapiens | |||
15. | ALA4575590 | 30 | EC50 | = | 0.061 | uM | ALA4478445 | 7.21 | nM | Human immunodeficiency virus 1 | ||
16. | ALA4575590 | 30 | IC50 | = | 0.033 | uM | ALA4478444 | 7.48 | nM | Human immunodeficiency virus 1 | ||
17. | ALA4575590 | 30 | Activity | = | 100 | % | ALA4478442 | % | Human immunodeficiency virus 1 | |||
18. | ALA4575590 | 30 | Activity | = | 100 | % | ALA4478443 | % | Homo sapiens |